Tianeptine

Tianeptine (brand names Stablon, Coaxil, Tatinol, Tianeurax and Salymbra) is a drug used primarily in the treatment of major depressive disorder, although it may also be used to treat asthma or irritable bowel syndrome. Chemically it is a tricyclic antidepressant (TCA), but it has different pharmacological properties than typical TCAs as recent research suggests that tianeptine produces its antidepressant effects through indirect alteration of glutamate receptor activity (i.e., AMPA receptors and NMDA receptors) and release of BDNF, in turn affecting neural plasticity.

Tianeptine has antidepressant and anxiolytic (anti-anxiety) properties with a relative lack of sedative, anticholinergic and cardiovascular adverse effects, thus suggesting it is particularly suitable for use in the elderly and in those following alcohol withdrawal; such persons can be more sensitive to the adverse effects of psychotropic drugs. Recent results indicate possible anticonvulsant (anti-seizure) and analgesic (painkilling) activity of tianeptine via immediate or downstream modulation of adenosine A1 receptors (as the effects could be experimentally blocked by antagonists of this receptor).

Tianeptine is a low-affinity full agonist at the μ-opioid and δ-opioid receptors with negligible effect at the κ-opioid receptors. μ-Opioid agonists typically induce euphoria, and in accordance, tianeptine does so at high doses well above the normal therapeutic range.

Product Introduction: 

Place of orgin: China

Specification:

1.Product name:Tianeptine

2.CAS No.:66981-73-5

3.Purity: 99% min

Synonyms:View MoreCOAXIL; Tianeptina; Tianeotine; Tianeptinum; Tianeptine-d4; Tianeptineacid; Tianeptina [inn-spanish]

Storage information: Store in Cool and dry .place, keep away from strong light, high temperature

Usage: intermediate,fine chemical

Transportation：by air express delivery(DHL,FedEx,EMS ect.) or sea shipping (FOB,CIF,CFR,CNF ect.)

Sample：sample can be supplied if you inquiry 

Price: we will give you the best price!

Specification:

Packaging & Shipping

Packing:1:We adopt different packing methods,According to the product .

                      Poly Bag Inner, Woven Bag outer,kraft paper bags,

                      Fibra bag or Drum and so on.

                 2:According to customer's requirement!

Shipping:We supply different transportations.

                   International courier like(TNT UPS DHL FEDEX)

                   We also supply by Air,by Sea

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Notice: This product is only suitable for laboratory use, or the use of animals. It can not be used directly on the human body